An Atom Economic Acid Catalyzed Synthetic Method for Aromatic Imines
نویسندگان
چکیده
منابع مشابه
Aza-pinacol rearrangement: acid-catalyzed rearrangement of aziridines to imines.
A series of di-, tri-, and tetra-substituted N-tosylaziridines [N-(toluene-p-sulfonyl)aziridines] 1, prepared by aziridination of the corresponding alkenes with N-[(tolyl-p-sulfonyl)imino]phenyliodinane (TsN = IPh), was found to undergo a BF3-catalyzed rearrangement (aza-pinacol rearrangement) under mild conditions to give the corresponding N-tosylimines 2 generally in satisfactory yields.
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ژورنال
عنوان ژورنال: Asian Journal of Chemistry and Pharmaceutical Sciences
سال: 2017
ISSN: 2456-6217
DOI: 10.18311/ajcps/2017/10991